CAS RN 1619994-68-1
IUPAC Navn:
1-[1-(2-methanesulfonylphenyl)-7-propoxyindolizin-3-yl]ethan-1-one
Synonymer:
1-[1-(2-methanesulfonylphenyl)-7-propoxyindolizin-3-yl]ethanone
Molekylvægt (g/mol):
371.45
Molekylformel:
C20H21NO4S
InChi Key:
KHWCPNJRJCNVRI-UHFFFAOYSA-N
SMILES:
CCCOC1=CC2=C(C=C(N2C=C1)C(C)=O)C1=CC=CC=C1S(C)(=O)=O
1
–
2
af
2
Resultater
2
GSK2801, MedChemExpress
MedChemExpress GSK2801 is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with Kd values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4.