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Tocris Bioscience™ Selpercatinib
Potent and selective RET inhibitor
1455.00 DKK - 5425.00 DKK
Specifications
| Chemical Name or Material | 6-(2-Hydroxy-2-methylpropoxy)-4-[6-[6-[(6-methoxy-3-pyridinyl)methyl]-3,6-diazabicyclo[3.1.1 ]hept-3-yl]-3-pyridinyl]pyrazolo[1,5-a]pyridine-3-carbonitrile |
|---|---|
| CAS | 2152628-33-4 |
| Target | Ret |
| Molecular Formula | C29H31N7O3 |
| Purity | 0.98 |
| Product Code | Brand | Quantity | Price | Quantity & Availability | |||||
|---|---|---|---|---|---|---|---|---|---|
| Product Code | Brand | Quantity | Price | Quantity & Availability | |||||
|
18747026
|
Tocris Bioscience™
7696/10 |
10 mg |
1455.00 DKK
10mg |
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|
18759196
|
Tocris Bioscience™
7696/50 |
50 mg |
5425.00 DKK
50mg |
Please sign in to purchase this item. Need a web account? Register with us today! | |||||
Description
Selpercatinib, is a potent and selective receptor tyrosine kinase RET inhibitor (EC50 = 4 nM). It shows > 100-fold selectivity for > 95% of 228 purified kinase domains in radiometric assays. In vitro, it inhibits proliferation of cancer cell lines containing RET mutations or gene fusions. In vivo, it inhibits tumor growth in diverse RET mouse models. Selpercatinib is orally bioavailable.Specifications
| 6-(2-Hydroxy-2-methylpropoxy)-4-[6-[6-[(6-methoxy-3-pyridinyl)methyl]-3,6-diazabicyclo[3.1.1 ]hept-3-yl]-3-pyridinyl]pyrazolo[1,5-a]pyridine-3-carbonitrile | |
| Ret | |
| 0.98 |
| 2152628-33-4 | |
| C29H31N7O3 |
Safety and Handling
Recommended Storage : Store at -20°C
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Product Title
Tocris Bioscience™ Selpercatinib