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Tocris Bioscience™ Selpercatinib

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Quantity:
10 mg
50 mg
Unit Size:
10mg
50mg
Description
Selpercatinib, is a potent and selective receptor tyrosine kinase RET inhibitor (EC50 = 4 nM). It shows > 100-fold selectivity for > 95% of 228 purified kinase domains in radiometric assays. In vitro, it inhibits proliferation of cancer cell lines containing RET mutations or gene fusions. In vivo, it inhibits tumor growth in diverse RET mouse models. Selpercatinib is orally bioavailable.
Greener Choice Claims
- Environmental benefits include:
- Ozone-Safe or Safe for the Ozone Layer

Specifications
Specifications
Chemical Name or Material | 6-(2-Hydroxy-2-methylpropoxy)-4-[6-[6-[(6-methoxy-3-pyridinyl)methyl]-3,6-diazabicyclo[3.1.1 ]hept-3-yl]-3-pyridinyl]pyrazolo[1,5-a]pyridine-3-carbonitrile |
CAS | 2152628-33-4 |
Quantity | 10 mg |
Target | Ret |
Molecular Formula | C29H31N7O3 |
Purity | 0.98 |
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