CAS RN 171714-84-4

IUPAC Navn: —

Synonymer: —

Molekylvægt (g/mol): —

Molekylformel: —

InChi Key: —

SMILES: —

1 – 1 af 1 Resultater

Darusentan, MedChemExpress

MedChemExpress Darusentan (Lu-135252) is a selective endothelin receptor A (ET-A) receptor antagonist, which binds with a Ki of 1.4 nM to the ET-A receptor and a Ki of 184 nM to ET-B receptor, respectively with a 100-fold selectivity for ETA rather than ETB receptors. Darusentan competes for radiolabeled endothelin binding in rat aortic vascular smooth muscle cells (RAVSMs) membranes with single-site kinetics, exhibiting a Ki of 13 nM.

Pris og tilgængelighed
Tekniske data

Kemisk navn eller materiale	Darusentan
Sundhedsfare 1	H302∣H315∣H319∣H335
Formel vægt	410.42
Opløselighedsinformation	DMSO : 100 mg/mL (243.65 mM; Need ultrasonic)
Procent renhed	98.66%
Fysisk form	Solid
Farve	White
Grad	Research
Anbefalet opbevaring	Powder -20°C 3 years, 4°C 2 years∣In solvent -80°C 6 months, -20°C 1 month
Molekylvægt (g/mol)	410.42
CAS	171714-84-4
Synonym	Lu-135252
Holdbarhed	Powder -20°C 3 years, 4°C 2 years∣In solvent -80°C 6 months, -20°C 1 month
SMIL	COC1=NC(O[C@H](C(O)=O)C(C2=CC=CC=C2)(C3=CC=CC=C3)OC)=NC(OC)=C1
Renhedsgrad noter	Research
Molekylær formel	C₂₂H₂₂N₂O₆
Til brug med (applikation)	COVID-19-immunoregulation

CAS RN 171714-84-4

Filtrerede søgeresultater

Snævre resultater