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Darusentan, MedChemExpress

Artikelnummer. 16466488
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16466488 10 mg
16452587 50 mg
16429077 5 mg
16426756 100 mg
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Artikelnummer. 16466488 Leverandør Medchem Express Leverandørnr. HY15404

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Beskrivelse

MedChemExpress Darusentan (Lu-135252) is a selective endothelin receptor A (ET-A) receptor antagonist, which binds with a Ki of 1.4 nM to the ET-A receptor and a Ki of 184 nM to ET-B receptor, respectively with a 100-fold selectivity for ETA rather than ETB receptors. Darusentan competes for radiolabeled endothelin binding in rat aortic vascular smooth muscle cells (RAVSMs) membranes with single-site kinetics, exhibiting a Ki of 13 nM.

Darusentan (Lu-135252) is a selective endothelin receptor A (ET-A) receptor antagonist, which binds with a Ki of 1.4 nM to the ET-A receptor and a Ki of 184 nM to ET-B receptor, respectively with a 100-fold selectivity for ETA rather than ETB receptors. Darusentan competes for radiolabeled endothelin binding in rat aortic vascular smooth muscle cells (RAVSMs) membranes with single-site kinetics, exhibiting a Ki of 13 nM.

Tekniske data

Kemisk navn eller materiale Darusentan
Fysisk form Solid
CAS 171714-84-4
Farve White
Mængde 10 mg
Renhedsgrad noter Research
Molekylær formel C22H22N2O6
Til brug med (applikation) COVID-19-immunoregulation
Synonym Lu-135252
Opløselighedsinformation DMSO : 100 mg/mL (243.65 mM; Need ultrasonic)
SMIL COC1=NC(O[C@H](C(O)=O)C(C2=CC=CC=C2)(C3=CC=CC=C3)OC)=NC(OC)=C1
Molekylvægt (g/mol) 410.42
Formel vægt 410.42
Procent renhed 98.66%
Grad Research
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Research purposes only

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