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Inobrodib, MedChemExpress

Artikelnummer. 16474528
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16474528 10 mg
16420837 50 mg
16407247 5 mg
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Artikelnummer. 16474528 Leverandør Medchem Express Leverandørnr. HY111784

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Beskrivelse

MedChemExpress Inobrodib (CCS1477) is an orally active, potent, and selective inhibitor of the p300/CBP bromodomain. Inobrodib binds to p300 and CBP with Kd values of 1.3 and 1.7 nM, respectively, and with 170/130-fold selectivity compared with BRD4 with a Kd of 222 nM. CCS1477 inhibits cell proliferation in prostate cancer cell lines and decreases androgen receptor (AR)- and C-MYC-regulated gene expression.

Inobrodib (CCS1477) is an orally active, potent, and selective inhibitor of the p300/CBP bromodomain. Inobrodib binds to p300 and CBP with Kd values of 1.3 and 1.7 nM, respectively, and with 170/130-fold selectivity compared with BRD4 with a Kd of 222 nM. CCS1477 inhibits cell proliferation in prostate cancer cell lines and decreases androgen receptor (AR)- and C-MYC-regulated gene expression.

Tekniske data

Kemisk navn eller materiale Inobrodib
CAS 2222941-37-7
Farve Off-White
Renhedsgrad noter Research
Molekylær formel C30H32F2N4O3
Mængde 10 mg
Synonym CCS1477
Opløselighedsinformation DMSO : 100 mg/mL (187.06 mM; Need ultrasonic)
SMIL O=C1N(C2=CC=C(F)C(F)=C2)[C@H](C3=NC4=CC(C5=C(C)ON=C5C)=CC=C4N3[C@H]6CC[C@H](OC)CC6)CCC1
Molekylvægt (g/mol) 534.6
Formel vægt 534.6
Procent renhed 99.41%
Grad Research
Fysisk form Solid
Til brug med (applikation) Cancer-programmed cell death
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Research purposes only

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