missing translation for 'onlineSavingsMsg'
Få mere at vide
Få mere at vide
Tocris Bioscience™ Ro 31-8220 mesylate

Klik for at se tilgængelige muligheder
Mængde:
10 mg
Beskrivelse
Protein kinase C inhibitor, with activity at other protein kinases (IC50 values are 33, 3, 8, 15 and 38 nM for PKCα, MAPKAP-K1b, MSK1, GSK3β and S6K1 respectively). Activates JNK and glycogen synthase, and inhibits MAPK and ERK2, in rat adipocytes and L6 myotubes. Also inhibits voltage-dependent Na+ channels in the micromolar range. Induces protein-protein interaction between mutant SMAD4R361H and SMAD3, leading to reactivation of dormant SMAD4R361H-mediated transcriptional activity and restoration of TGF-β-induced tumor suppression activity in SMAD4 mutant cancer cells.
Tekniske data
Tekniske data
| Kemisk navn eller materiale | Ro 31-8220 mesylate |
| CAS | 138489-18-6 |
| Mængde | 10 mg |
| Molekylær formel | C26H27N5O5S2 |
| Formel vægt | 553.65 |
| Renhed | >97% |
| Molekylvægt (g/mol) | 553.652 |
Korrektion af produktindhold
Dit input er vigtigt for os. Udfyld denne formular for at give feedback relateret til indholdet på dette produkt.
Produkttitel
Ser du en mulighed for forbedring?Del en indholdskorrektion