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DiscoverX PathHunter™ eXpress c-KIT Functional Assay
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Mængde:
1.000 dp (10 x 96-brønds)
Beskrivelse
The PathHunter™ eXpress c-KIT Functional Assay provides an easy-to-use cell based assay to study drug candidates (small molecules or biologics) targeting RTKs. This kit assesses RTK activation via detection of activated c-KIT dimerization-induced SH2 domain protein recruitment. This product uses EFC technology. The included cells overexpress PK-tagged c-KIT and an EA-tagged SH2 domain protein. Upon ligand-induced receptor activation, SH2-EA recruitment leads to production of EFC signal. eXpress kits are a convenient, ready-to-use format which contains all materials needed to run the assay, including single-use vials of cryopreserved cells, cell plating media, detection reagent, and assay plates. Please note that this product expresses the Cyno version of the protein.
Tekniske data
Tekniske data
| Assay Entry | Receptor Phosphorylation |
| Til brug med (applikation) | Assay-Ready eXpress Kits |
| Primær agonist | Recombinant Human SCF |
| Mængde | 1.000 dp (10 x 96-brønds) |
| Målindgang | c-KIT |
| Cellelinje | U2OS |
| Mål | c-KIT |
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