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Tocris Bioscience™ I-BET 762

Artikelnummer. 18094322
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Mængde:
5 mg
25 mg
Denne vare kan ikke returneres. Se returpolicy

Artikelnummer. 18094322

Brand: Tocris Bioscience™ 6521/25

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Beskrivelse

Potent and high affinity BET bromodomain inhibitor; anti-inflammatory; orally bioavailable.

I-BET 762 is a potent and high affinity BET bromodomain inhibitor (IC50 = 32.5 - 42.5 nM; Kd = 50.5 - 61.3 nM). Inhibits myeloma cell proliferation. Attenuates transcription of oncogenic MYC and suppresses key inflammatory genes. Exhibits efficacy in a range of oncology and immunoinflammatory models. Displays antiproliferative effect in vitro and in vivo. Orally bioavailable.
TRUSTED_SUSTAINABILITY

Specifications

Kemisk navn eller materiale (4S)-6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide
CAS 1260907-17-2
Mængde 25 mg
Mål Bromodomain Inhibitors
Molekylær formel C22H22ClN5O2
Renhed 0.98
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