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Tocris Bioscience™ ERK5-IN-1

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Mængde:
10 mg
50 mg
Beskrivelse
ERK5-IN-1 is a potent and selective ERK5 inhibitor; inhibits EGFR-induced ERK5 autophosphorylation (EC50 = 90 nM) and ERK5 enzymatic activity (IC50 = 162 nM). Exhibits at least 30-fold selectivity for ERK5 over LRRK2 in a cell based assay. Also selective for ERK5 over a panel of other kinases. Orally bioavailable.
Tekniske data
Tekniske data
| Renhed | >98% |
| Oversigt | ERK5-IN-1 |
| Molekylvægt (g/mol) | 638.8 |
| Produkttype | ERK5-IN-1 |
| Mængde | 10 mg |
For Research Use Only
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